Vepafestinib
产品介绍
Vepafestinib是一种酪氨酸激酶抑制剂(TKI),潜在用于癌症治疗,特别是白血病或实体瘤。
产品性质
产品特色
/
存储条件
-25~-15℃避光保存,有效期3年。
COA
已发表文献
[1] Miyazaki I, Odintsov I, Ishida K, Lui AJW, Kato M, Suzuki T, Zhang T, Wakayama K, Kurth RI, Cheng R, Fujita H, Delasos L, Vojnic M, Khodos I, Yamada Y, Ishizawa K, Mattar MS, Funabashi K, Chang Q, Ohkubo S, Yano W, Terada R, Giuliano C, Lu YC, Bonifacio A, Kunte S, Davare MA, Cheng EH, de Stanchina E, Lovati E, Iwasawa Y, Ladanyi M, Somwar R. Vepafestinib is a pharmacologically advanced RET-selective inhibitor with high CNS penetration and inhibitory activity against RET solvent front mutations. Nat Cancer. 2023 Sep,4(9):1345-1361. doi: 10.1038/s43018-023-00630-y. Epub 2023 Sep 21. Erratum in: Nat Cancer. 2023 Oct,4(10):1526. doi: 10.1038/s43018-023-00663-3. PMID: 37743366, PMCID: PMC10518257.
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